Tlhaloso ea Sehlahisoa
Testosterone undecanoate Phofo Video-AASraw
Testosterone e tala undecanoate Powder Basic Characters
Name Product: | Testosterone e se nang phofo e ntle |
CAS: | 5949-44-0 |
Molecular Formula: | C30H48O3 |
Boima ba 'mele: | 456.71 |
Melt Point: | 59-61 ° C |
Assay: | 98% mets(HPLC) |
Temp Temp Storage: | -20 ° C Freezer |
Color: | Phosente e tšoeu ea kristale |
Testosterone undecanoate History le Overview
Testosterone undecanoate ke steroid ea nako e telele le e liehang ho lokolloa, e sebetsa e le prodrug ea testosterone, e lokelang ho nkoa e le mofuta oa tlhaho le oa tlhaho oa testosterone, o ka arabela bakeng sa khōlo e tloaelehileng le nts'etsopele ea litho tsa botona kapa botšehali tsa banna. E qalile ho sebelisoa bakeng sa tšebeliso ea bongaka ho phekola testosterone e tlaase ka Schering AG, in1954.E amoheloa ke US Food and Drug Administration (FDA), ngaka e tla fana ka eona e le Testosterone Replacement Therapy (TRT), kapa maemo a mang (a kang: kankere ea tšoelesa ea senya, ho lahleheloa ke boima ba 'mele, le ho se sebetse hantle ka thobalano). Kaha testosterone ea eona e 'nile ea kenngoa le ester ea undecanoate sehlopheng sa 17-beta hydroxyl, se nang le phapang e kholo ho tse ling tsohle tsa oral anabolic steroids kaha ha li na methylation (C-17 alpha alkylation) ka carbon 17th. Kahoo, testosterone undecanoate ha e hlahise liphello tse mpe sebeteng joaloka metsoako ea C-17 alpha alkylated. Ntle le moo, matla a Testosterone undecanoate le nako e telele ea ts'ebetso, e ka kena 'meleng ka lymphatic system ka pampitšana ea GI, ea kenngoa habonolo' meleng, hangata ke lithethefatsi tse ratoang tsa kalafo bakeng sa maemo a tlase a Testosterone.
Testosterone undecanoate Powder ke eng?
Testosterone undecanoate e qalile ho rekisoa le ho ajoa Inthaneteng bakeng sa merero ea bongaka ka fektheri ea eona, moetsi, mofani oa thepa, haholo-holo e hlaha ka mefuta e 'meli e nang le ente le ea molomo tlas'a lebitso la eona "Andriol, Aveed, Understor le Nebido har'a ba bang' marakeng ona, hape o bitsoa "testosterone". undecylate, test undecanoate, test u, TU, joalo-joalo. ”.
Testosterone undecanoate phofo ke ester e telele ea testosterone eo haholo-holo e sebelisang ho tšoara maemo a tlaase a Testosterone ho banna. Ho sa le joalo, e sebelisoa haholo ke baatlelete le baetsi ba 'mele ho ntlafatsa ts'ebetso ea motho ka kakaretso. Ka lebaka la halofo ea nako e telele ea bophelo, phofo ea testosterone undecanoate ha e hloke tsamaiso ea kamehla. Ka lebaka la sena, liphello tsa eona tse ntle li ka lieha haholo 'me li ka' na tsa se ke tsa qala ho thusa ho fihlela qetellong ea potoloho e tloaelehileng ea steroid. E lumellana hantle le lipotoloho tsohle le merero ea ts'ebetso, e ka ntlafatsa tsebo ea bona ea ho aha 'mele le ts'ebetso ea thobalano ka kakaretso, hape e ka ba thusa ho fumana mesifa le ho lahleheloa ke mafura a' mele. Ka lebaka la ts'ebetso ea eona e potlakileng ea ketso le nako e telele ea halofo ea bophelo 'meleng, phofo ea testosterone undecanoate hangata e nkoa e sebetsa ho feta. testosterone cypionate le testosterone enanthate. Ha ho bapisoa le mefuta ena e meng ea testosterone, theko e boetse e theko e tlaase.
Ke phello efe ea Testosterone undecanoate phofo sebetsa mmeleng wa hao
Testosterone undecanoate phofo ke mafura a mafura a nako e telele a kenngoa hantle 'meleng ka mala a manyenyane, ebe o kenngoa ka har'a sebete ho fetola testosterone. Ha testosterone ena e kena maling, e tla e kopanya le li-receptor tsa androgen, tse fumanoang liseleng tsa mesifa. Hang ha testosterone e tlama ho li-receptor tsena, e susumetsa protheine synthesis le kholo ea mesifa. Testosterone undecanoate phofo ke steroid e sebetsang butle-butle e le halofo ea nako e telele haholo ea bophelo, e hloka nako e telele ho boloka boemo bo botle ba ho lula tsamaisong, joale e ka laola ho lokolloa ha hormone 'meleng. Kahoo, baetsi ba 'mele ba bangata le baatlelete ba reka phofo ea Testosterone undecanoate ho ntlafatsa ponahalo ea bona ea' mele le matla a bona ka kakaretso.
Mokhoa oa ho sebelisa Testosterone e se nang phofo e ntle Bakeng sa ho haha 'mele
(1)Testosterone e se nang phofo e ntle tekanyo
Pele o qala ho sebelisa testosterone undecanoate phofo, ke habohlokoa ho tseba tekanyo e nepahetseng le potoloho. Tekanyo ea phofo ea Testosterone undecanoate e fapana ho itšetlehile ka motho ka mong le lipakane tsa bona. Tekanyo e tloaelehileng e pakeng tsa 80 mg le 160 mg ka letsatsi; qala ka tekanyo e tlase 'me butle-butle u e phahamise ho fumana tekanyo e nepahetseng; pheta potoloho ena libeke tse ling le tse ling tse 4-6; ’me u e nke ka nako e tšoanang letsatsi ka leng kapa ka ntle ho lijo.
(2)Testosterone e se nang phofo e ntle bolelele ba potoloho
Testosterone undecanoate phofo ha se sehlahisoa sa testosterone se ratoang haholo, se hloka ho sebelisoa ka tekanyo e phahameng bakeng sa baetsi ba 'mele le baatlelete ho fumana ts'ebetso kapa ntlafatso ea' mele ka potoloho ea boinotšing ka lebaka la ho fokotseha ha eona ka bioavailability. Leha ho le joalo, liphetho tsa potoloho ea phofo ea testosterone undecanoate bakeng sa ho aha 'mele hangata li utloahala li koaletsoe hantle ka li-anabolic steroids tse ling (joalo ka: winstrol, anavar kapa nandrolone) ho fihlela litlamorao tsa potoloho ea eona. E kanna ea nka nako e telele ho feta lipotoloho tse tloaelehileng ka lebaka la sebopeho sa eona sa ho sebetsa butle, empa e ka thusa ho fihlela sepheo se nepahetseng sa boikoetliso. Joalokaha re tseba hore, testosterone undecanoate phofo ke mofuta o tsitsitseng oa testosterone o sa hlahiseng litla-morao tsa estrogenic, e 'nile ea bontšoa ho hlahisa mesifa le matla a mangata ho feta. testosterone enanthate kapa testosterone cypionate.
(3)Testosterone e se nang phofo e ntle halofo ea bophelo
Ho itšetlehile ka potoloho, halofo ea bophelo ea Testosterone Undecanoate phofo ke 3 ho lihora tsa 7.
(4)Testosterone e se nang phofo e ntle liphetho bakeng sa bodybuilding
Testosterone undecanoate powder ke ester e sebetsang butle e hlokang potoloho e telele ho fumana liphello tse atlehang, haeba u ka rata ho reka phofo ea Testosterone undecanoate Inthaneteng e le lithethefatsi tse ntlafatsang ts'ebetso, steroid ena ka sebele e ka tlisa melemo e mengata bakeng sa baetsi ba 'mele kapa basebelisi ba ts'ebetso. , tsena li kenyelletsa:
'Misa oa mesifa o eketsehileng: Testosterone undecanoate phofo ke hormone ea bohlokoa bakeng sa ho hōla ha mesifa, e ka khothalletsa kholo e kholo ea mesifa le nts'etsopele ka ho eketsa litekanyetso tsa testosterone
Matla le Matla a Eketsehileng: Nka testosterone undecanoate phofo e le tlatsetso e ka bona keketseho e kholo ea matla le matla. Sena se ka ba molemo ho baatlelete le baetsi ba 'mele ba hlokang ho sebetsa ka hohle kamoo ba ka khonang ka nako e telele.
Maemo a Fokotseng a Mafura: Testosterone undecanoate phofo e ka fokotsa maemo a mafura, ho thusa ho theola boima ba 'mele le ho finyella' mele o fokolang.
Linako tse Ntlafetseng tsa ho Pholosa: Testosterone undecanoate phofo e ka thusa baatlelete le baetsi ba 'mele hore ba hlaphoheloe ka potlako ho tloha ho ikoetlisa ka matla.
Kotsi e fokotsehileng ea kotsi: Testosterone undecanoate phofo e ka fokotsa kotsi ea kotsi ka ho thusa mesifa ho lokisa tšenyo ka potlako. Ka lebaka leo, baatlelete ha ba na monyetla oa ho khathala kapa ho tsoa likotsi nakong ea boikoetliso.
Testosterone undecanoate Pkolota Phekolo ea Post-Cycle Therapy(PCT)
Tlhahiso ea tlhaho ea testosterone 'meleng oa hau e tla hatelloa ka ho sebelisa phofo ea testosterone undecanoate, tekanyo ea khatello ena e tla itšetleha ka tekanyo ea phofo ena le lintho tse ling tse sebelisoang ho pholletsa le potoloho ea hau. Ho tsosolosoa ha maemo a testosterone a tlhaho ho ka thusoa ke phekolo ea post-cycle. Ho khutlisetsa 'mele oa hau maemong a tloaelehileng qetellong ea potoloho, PCT e bohlokoa. Ho etsa PCT, o ka sebelisa li-supplement tse fapaneng joalo ka Clomid, Nolvadex, le HCG. Khetha e le 'ngoe kapa tse peli ho tsena ho nka libeke tse' nè, ebe butle-butle fokotsa tekanyo ho litlhoko tsa hau.
Mekhoa e meng ea eona ho Testosterone undecanoate Powder
Testosterone undecanoate phofo e ka kenngoa ka mekhoa e mengata ea tlhaho ho finyella lipakane tse itseng tsa ho haha 'mele, tse latelang ke tse ling tse tloaelehileng:
Bulking stack: Testosterone undecanoate, Dianabol, le HGH
Ho khaola stack: Testosterone undecanoate, Winstrol, le Clenbuterol
Matla a stack: Testosterone undecanoate, Trenbolone, le Deca Durabolin
Endurance stack: Testosterone undecanoate, Anavar, le Creatine
Recovery stack: Testosterone undecanoate, BCAAs, le glutamine
Le hoja mofuta o mong le o mong oa testosterone replacement therapy (TRT) o na le melemo le likotsi tsa oona, kaofela ha tsona li ikemiselitse ho phahamisa maemo a testosterone ka maiketsetso ha li ntse li fokotsa kotsi ea litla-morao le ho phahama ha khatello ea mali. Ka lebaka leo, ho bohlokoa ho buisana le ngaka pele u qala mefuta e meng ea tlhaho.
Ke eng Testosterone undecanoate Pkolota phello e lehlakoreng
Testosterone undecanoate e nkoa e le phekolo e sireletsehileng le e sebetsang ea testosterone (TRT), empa basebelisi ba ka 'na ba e-ba le litla-morao tse ka' nang tsa e-ba teng haeba ba sa tsebe ho li sebelisa kapa ho sebelisa hampe testosterone undecanoate phofo le potoloho, tsena li kenyelletsa:
▪ Mokhathala
▪ Ho hlobaela
▪ Ho feto-fetoha ha maikutlo
▪ Ho eketseha ha boima ba ’mele
▪ Eketsa Lehloba
▪ Ho opeloa sebakeng sa ente
▪ Lefatla (Ho hlotheha ha Moriri)
▪ Gynecomastia
▪ Hypogonadism
▪ Khatello ea mali
▪ Keketseho ea estradiol
▪ Li-enzyme tse phahameng tsa sebete
▪ Hypertriglyceridemia
▪ Kotsi ea virilization (Basebelisi ba basali)
▪ Moriri oa 'mele oa hola (Basebelisi ba basali)
▪ Lentsoe le tebileng (Basebelisi ba basali)
Lethathamo le ka holimo leha e le efe ea matšoao ana ao u nang le 'ona, ka kopo emisa ho sebelisa phofo ea testosterone undecanoate pele, kaha boholo ba litla-morao tsena ke tsa nakoana, li tla rarolla ka bobona. Ka kopo tsebisa ngaka ea hau hang-hang haeba u tsoela pele ho ba le matšoao ana kapa haeba a mpefala ha nako e ntse e ea.
Ke mohloli ofe o bolokehileng ho reka Testosterone undecanoate Phofo?
Testosterone Undecanoate phofo e 'nile ea bontšoa e sireletsehile le e sebetsang bakeng sa ho ntlafatsa liphello tsa ho haha' mele, e ka thusa ho eketsa boima ba mesifa, matla le mamello, ha e ntse e ka fokotsa mafura a 'mele. Ke e 'ngoe ea li-supplement boosting tse ratoang ka ho fetisisa tšimong ea ho haha' mele, maikutlo a mangata a matle a ka bonoa ho baetsi ba 'mele ba sebelisitseng steroid ena. Haeba u rerile ho laela phofo e hloekileng ea testosterone undecanoate inthaneteng, websaeteng e nang le botumo bo botle ba steroid e tla ba khetho e ntle haholo.
AASraw ke moetsi ea hloahloa oa testosterone undecanoate powder e nang le lab e ikemetseng le fektheri e kholo e le ts'ehetso, tlhahiso eohle e tla etsoa tlas'a taolo ea CGMP le tsamaiso ea tsamaiso ea boleng bo sebetsang. Tsamaiso ea phepelo e tsitsitse, testosterone undecanoate phofo e ngata ea thekiso le litaelo tse ngata li amoheleha.
Tlaleho e Raw Testosterone undecanoate Powder Testing-HNMR
HNMR ke eng hona HNMR spectrum e u bolella eng? H Nuclear Magnetic Resonance (NMR) spectroscopy ke mokhoa oa ho hlahloba k'hemistri o sebelisoang ho laola boleng le lipatlisiso bakeng sa ho fumana likahare le bohloeki ba sampuli hammoho le sebopeho sa limolek'hule. Mohlala, NMR e ka sekaseka ka bongata metsoako e nang le metsoako e tsebahalang. Bakeng sa metsoako e sa tsejoeng, NMR e ka sebelisoa ho bapisa le lilaebrari tsa spectral kapa ho fana ka sebopeho sa motheo ka kotloloho. Hang ha sebopeho sa motheo se tsejoa, NMR e ka sebelisoa ho fumana hore na limolek'hule li lumellana joang le tharollo hammoho le ho ithuta thepa ea 'mele boemong ba limolek'hule joalo ka phapanyetsano ea conformational, liphetoho tsa mohato, solubility le diffusion.
Testosterone Undecan0ate (5949-44-0) -COA
Testosterone Undecanate phofo (5949-44-0) -COA
Joang ho reka Testosterone undecanoate Phofo e tsoang ho AASraw?
❶Ho ikopanya le rona ka mokhoa oa rona oa ho botsa ka lengolo-tsoibila, kapa ho re siela nomoro ea hau ea WhatsApp, moemeli oa rona oa litšebeletso tsa bareki (CSR) o tla ikopanya le uena ka mor'a lihora tse 12.
❷ Ho re fa palo le aterese eo u e botsitseng.
❸ CSR ea rona e tla u fa khotheishene, nako ea ho patala, nomoro ea ho sala morao morao, mekhoa ea ho fihla le letsatsi la ho fihla (ETA).
❹Ho lefa 'me thepa e tla romelloa ka mor'a lihora tse 12.
❺Lintho tse amohetsoeng le ho fana ka maikutlo.
Mongoli oa sengoloa sena:
Ngaka Monique Hong o fumane lengolo UK Imperial College London Faculty of Medicine
Sengoli sa pampiri sa Scientific Journal:
1. Mathias Hallberg
The Beijer laboratory, Department of Pharmaceutical Biosciences, Neuropharmacology and Addiction Research, Uppsala University, SE-751 24, Sweden
2. Marc Gittelman MD
Lefapha la Urology, Sekolo sa Bongaka sa Univesithi ea New York, New York, NY, USA
3. Jeffrey D. Freid MD
Karolo ea Urology, Lefapha la Ho Buoa, Univesithi ea Utah School of Medicine, Salt Lake City, UT, USA
4. Stefan M. Pasiakos
Karolo ea Phepo ea Sesole, Setsi sa Lipatlisiso sa Sesole sa US sa Meriana ea Tikoloho, Natick, MA, USA
Ha ho ka tsela leha e le efe ngaka/saense ena e buellang kapa ho buella ho rekoa, thekiso, kapa tšebeliso ea sehlahisoa sena ka lebaka lefe kapa lefe. Aasraw ha e na kamano kapa kamano, ho boleloa kapa ho seng joalo, le ngaka ena. Sepheo sa ho qotsa ngaka ena ke ho ananela, ho ananela le ho babatsa lipatlisiso tse felletseng le mosebetsi oa nts'etsopele o entsoeng ke bo-ramahlale ba sebetsanang le ntho ena.
Reference
[1] Corona, G., Maseroli, E., & Maggi, M. (2014). Testosterone e nang le ente ea undecanoate bakeng sa kalafo ea hypogonadism. Maikutlo a Setsebi ka Pharmacotherapy, 15(13), 1903-1926. doi: 10.1517/14656566.2014.944896.
[2] Köhn FM, Schill WB (November 2003). "Tekanyetso e ncha ea molomo ea testosterone undecanoate". Journal ea Lefatše ea Urology. 21 (5): 311–315. doi:10.1007/s00345-003-0372-x. PMID 14579074.
[3] Testosterone Undecanoate-Schering AG. Lithethefatsi ho R&D. 5 (6): 368–369. 2004. doi:10.2165/00126839-200405060-00012. PMID 15563244.
[4] Jacobeit JW, Gooren LJ, Schulte HM (Lwetse 2007). "Testerone undecanoate ea nako e telele ea intramuscular bakeng sa kalafo ea batho ba transgender ea basali ho ea ho banna". Journal of Sexual Medicine. 4 (5): 1479–1484. doi:10.1111/j.1743-6109.2007.00556.x. PMID 17635694.
[5] Ong GS, Somerville CP, Jones TW, Walsh JP (2012). "Anaphylaxis e bakoang ke benzyl benzoate ha ho etsoa depo testosterone undecanoate". Litlaleho tsa Nyeoe ho Meriana. 2012: 384054. doi:10.1155/2012/384054. PMC 3261473. PMID 22272209. 384054.
[6] Behre HM, Abshagen K, Oettel M, Hübler D, Nieschlag E (May 1999). "Intramuscular ente ea testosterone undecanoate bakeng sa phekolo ea hypogonadism ea banna: lithuto tsa mohato oa pele". European Journal of Endocrinology. 140 (5): 414–419. CiteSeerX 10.1.1.503.1752. doi:10.1530/eje.0.1400414. PMID 10229906.
[7] Ke li-hormone life tse sebelisoang hangata bakeng sa phetisetso ea thobalano ea litlhapi (Bolaoli)